Compound Target Indication (Combination) Stage of Development Partner
Clinical Programs - IAP Platform
HGS1029 Inhibitor of Apoptosis Proteins (IAPs) Solid Tumors Phase I
Preclinical Programs
IAP Inhibitors Inhibitor of Apoptosis Proteins (IAPs) Inflammation/autoimmune Optimized Lead Compounds  
Tyrosine Kinase Inhibitors • BTK
• FMS
Inflammation/autoimmune, Oncology Early Lead Compounds  
HSP90 Inhibitors HSP90 Fungal Infections, CNS, Inflammation, Oncology Early Lead Compounds